Logo image
Counterattack reagent bis(trimethylsilyl)acetamide in the disilylation of diols
Journal article   Peer reviewed

Counterattack reagent bis(trimethylsilyl)acetamide in the disilylation of diols

Jih Ru Hwu, Denise A. Anderson, Naelong Wang, Meredith M. Buchner, Paul Gani and Shwu‐Chen Tsay
Chemische Berichte, Vol.123(8), pp.1667-1671
1990

Abstract

Bis(trimethylsilyl)acetamide Counterattack reagent Diol Disilylation Tandem doublecounterattack process
The counterattack method was applied to the disilylation of diols. Treatment of various diols with 0.3 or 1.1 equivalents of potassium hydride and 1.1 equivalents of bis(trimethylsilyl)‐acetamide in THF gave the corresponding disilyl ethers in good to excellent yields (60–95%). The diols may contain other functionalities, such as amide, amine, ether, and thioether. The diols used in the disilylation were 2a–14a. The newly developed disilylation proceeded in one flask by a sequential deprotonation‐silylation‐deprotonation‐silylation pathway. This disilylation also represents an example of a “tandem double‐counterattack process”. Bis(trimethylsilyl)‐acetamide acted as a counterattack reagent; it provided two Me 3 Si groups to diols and produced amides as bases. Copyright © 1990 WILEY‐VCH Verlag GmbH & Co. KGaA, Weinheim

Metrics

1 Record Views

Details

Logo image