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Gold-catalyzed dealkoxylative carbocyclization/[3+3] annulation cascade of acetal-allene or ketal-allene substrates
Journal article   Peer reviewed

Gold-catalyzed dealkoxylative carbocyclization/[3+3] annulation cascade of acetal-allene or ketal-allene substrates

Tse-Min Teng, Ming-Shiun Lin, Dhananjayan Vasu, Sabyasachi Bhunia, Ting-An Liu and Rai-Shung Liu
Chemistry - A European Journal, Vol.16(16), pp.4744-4748
26/04/2010

Abstract

Alienes Annulation Carbocyclization Cascade reactions Gold
(Chemical Equatation Reprentation) Rapid construction: We report the first successful implementation of a catalytic tandem carbocyclization/annulation cascade reaction (e.g., see scheme) using acetal-allene or ketal-aliene substrates through a dealkoxylative mode. This gold catalysis enables a rapid stereocontrolled construction of oxacyclic or carbocyclic frameworks. © 2010 Wiley-VCH Verlag GmbH & Co. KGaA,.

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