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Gold-catalyzed oxidative cycloadditions to activate a quinoline framework
Journal article   Peer reviewed

Gold-catalyzed oxidative cycloadditions to activate a quinoline framework

Deepak B. Huple, Satish Ghorpade and Rai-Shung Liu
Chemistry - A European Journal, Vol.19(39), pp.12965-12969
23/09/2013

Abstract

catalysis cycloaddition gold oxidative cyclization stereoselectivity
Going for gold! Gold-catalyzed reactions of 3,5- and 3,6-dienynes with 8-alkylquinoline oxides results in an oxidative cycloaddition with high stereospecificity (see scheme; EWG = electron-withdrawing group); this process involves a catalytic activation of a quinoline framework. The reaction mechanism involves the intermediacy of α-carbonyl pyridinium ylides (I) in a concerted [3+2]-cycloaddition with a tethered alkene. Copyright © 2013 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim.

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