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Stereocontrolled synthesis of functionalized bicyclic α-methylene butyrolactones via tungsten-mediated intramolecular allylation of aldehydes
Journal article   Peer reviewed

Stereocontrolled synthesis of functionalized bicyclic α-methylene butyrolactones via tungsten-mediated intramolecular allylation of aldehydes

Lin-Hun Shiu, Yang-Lian Li, Chien-Le Li, Ching-Yu Lao, Wei-Chen Chen and Rai-Shung Liu
Journal of Organic Chemistry, Vol.64(20), pp.7552-7558
01/10/1999

Abstract

The syntheses of a series of CpW(CO) 2 (π-γ-lactonyl) complexes bearing a tethered aldehyde are described. These π-allyl complexes are prepared as either syn- or anti-stereoisomers. Treatment of these dicarbonyl complexes with NOBF 4 and NaI in CH 3 CN effects an intramolecular allylation of the tethered aidehyde, yielding bicyclic α-methylene butyrolactones comprising a homoallylic alcohol. Both syn- and anti-isomers of tungsten-π-allyl compounds produce the same α-methylene butyrolactones. The cyclizations proceed with high diastereoselectivities to give only the cis-fused bicyclic γ-lactones. The preference for cis-fused stereoselection can be rationalized based on a tricyclic transition state mechanism.

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