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Substituent Effect on the Chlorination of 2-Alkoxypyridines to give 2-Chloropyridines under Vilsmeier-Haack Conditions
Journal article   Peer reviewed

Substituent Effect on the Chlorination of 2-Alkoxypyridines to give 2-Chloropyridines under Vilsmeier-Haack Conditions

Long-Li Lai, Pen-Yuan Lin, Jy-Shih Wang, Jih Ru Hwu, Min-Jen Shiao and Shwu-Chen Tsay
Journal of Chemical Research - Part S, (4), pp.194-195
04/1996

Abstract

Various substituted 2-alkoxypyridines were converted into the corresponding 2-chloropyridines in 28-91% yields by use of POCl 3 and DMF, in which the methyl, halogen, ester and nitro groups displayed an activating effect; in contrast, an amino group exhibited a deactivating effect.

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